Synthesis of quinazolinimines and quinazolinamines from 2-fluorobenzonitriles under catalyst-free conditions.
نویسندگان
چکیده
A convenient procedure for the synthesis of quinazolinimines and quinazolinamines from 2-fluorobenzonitriles has been developed. By using KO(t)Bu as the promotor with 2-aminopyridines or amidines as the reaction partner, the desired heterocycles were produced in moderate to good yields under catalyst-free conditions.
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 13 43 شماره
صفحات -
تاریخ انتشار 2015